Software Developed by the Donald Lab
OSPREY 3.0
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Welcome to the website for the OSPREY (Open Source
Protein REdesign
for You) software.
OSPREY is free and open-source software, and is available on Github, where you can always
find our latest updates. Please read
the licensing and legal terms first!
Please e-mail us if you have any questions.
The latest version of OSPREY is
3.2.101. It is significantly refactored compared to previous releases, and comes with
a convenient Python interface, as well as several new algorithms and marked performance improvements
including (but not limited to) GPU acceleration.
OSPREY is a suite of programs for computational structure-based protein design. OSPREY is developed in the lab of Prof. Bruce Donald at Duke University.
OSPREY is specifically designed to predict protein mutants that possess desired target properties (e.g., improved stability, switch of substrate specificity, etc.). OSPREY can also be used for predicting small-molecule drug inhibitors. Starting with version 2.0, OSPREY can now design protein-protein and protein-peptide interactions.
OSPREY incorporates several different algorithmic modules for
structure-based protein design, including a number of powerful
Dead-End Elimination algorithms and the ensemble-based K* algorithm
for protein-ligand binding prediction. OSPREY allows the incorporation
of continuous protein side-chain and continuous or discrete backbone
flexibility, while maintaining provable guarantees with respect to the
input model (input structure, rotamer library, energy function, and any backbone perturbations)
for a given protein design problem.
To our knowledge, OSPREY is the only open-source, freely-available
implementation of the DEE/A* algorithms. DEE/A* combines the provable
Dead-End Elimination (DEE) algorithms with the A* search
enumeration. OSPREY also includes many extensions and improvements to
the DEE framework (e.g., minDEE, iMinDEE, K*, DACS, BD, BRDEE, DEEPer, EPIC, COMETS, BWM*, LUTE, BBK*, and CATS). These
extensions improve efficiency and allow the modelling of molecular
flexibility. OSPREY includes the K* (pronounced "K-star") module,
which is a provably-good ε-approximation (epsilon-approximation)
algorithm for computing binding constants (KD) over
molecular ensembles of the bound and unbound states of a
protein:ligand complex using minimized DEE/A* (namely, minDEE/A*/K*).
See our papers for
details.
Legal Terms, Citation Requirements and Software License
To use Osprey, please first read the
following Citation
Requirements. In short, users must cite Osprey in papers,
patents, or presentations, and must use the name "Osprey" in the
text thereof.
Beyond that, OSPREY is free software and can be redistributed and/or
modified under the terms of version 2 of the GNU General Public
License as published by the Free Software
Foundation. OSPREY is distributed in the hope that it will be useful, but WITHOUT ANY WARRANTY; without even the implied warranty of MERCHANTABILITY or FITNESS FOR A
PARTICULAR PURPOSE. See the GNU General Public License for more details. Full licensing details, including citation requirements for the various different modules of
the software, are found on our Github page.
In particular, we require that everyone who publishes or presents results from OSPREY
to mention the name OSPREY and (if they used OSPREY 3) to cite our paper
introducing OSPREY 3.0, along with the papers for the specific
modules or algorithms they used
(see Github and/or below).
Examples and Bibliography
Selcted Examples and use-cases:
- Textbook
- Anti-infectives: Pathogen Resistance and Inhbitor
Resilience (Durability)
- Anti-neoplastics: Predicting
resistance mutations
- Anti-infectives: Predicting
resistance mutations (1)
- Anti-infectives: Predicting
resistance mutations (2)
- Anti-virals: Here is a tutorial by Brian Cox, on Osprey-based prediction of
influenza resistance mutations:
- Anti-neoplastics: T. Kaserer and J. Blagg.
Osprey-based workflow
predicts mutations likely to arise
upon drug treatment in a particular cancer tumor type.
- Antibodies: Design of biologics
- Computational
design of a tight binder to KRas, an "undruggable" cancer target, and
redesign of the Ras:Raf protein:protein interface
- Osprey-based Analysis of Energy Landscapes
- GPU
support, PPI design, Benchmarks, Advanced algorithms
- Tutorial
on Protein Design
- Multi-state
design and resistance mutations
Selected Empirical Designs that used OSPREY:
- Improved HIV-1 Neutralization Breadth and Potency of V2-Apex
Antibodies by In Silico Design (with G. Holt, J. Gorman,
S. Wang, A. Lowegard, B. Liu, T. Lin, B. Zhang, M. Louder,
M. Frenkel, K. McKee, S. Rawi, O'Dell R., C.-H. Shen, N. Doria-Rose,
and P. Kwong). Cell Reports (2023) In press.
- Discovery,
characterization, and redesign of potent antimicrobial thanatin
orthologs from Chinavia ubica and Murgantia
histrionica targeting E. coli LptA
(with K. Huynh,
A. Kibrom and P. Zhou). Journal of Structural Biology: X.
(2023) In press.
- Protocol for predicting drug-resistant protein mutations to an ERK2 inhibitor using RESISTOR
(with N. Guerin and T. Kaserer).
Cell STAR (Structured Transparent Accessible Reproducible)
Protococols 2023; 4(2):102170. doi: 10.1016/j.xpro.2023.102170.
-
RESISTOR: An algorithm for predicting
resistance mutations using Pareto optimization over multistate
protein design and mutational signatures
(with N. Guerin
and
T. Kaserer).
Journal: Cell Systems 2022; (13)10:
830-843 [PDF,
at journal],
and
Video
from Conference: RECOMB (May, 2022), San Diego.
- Non-canonical inhibitors target the CAL binding site: new
approaches to stabilize functional ΔF508-CFTR (with N. Gill,
J. Amacher, P. Cushing, Y. Zhao, L. Wallace, A. Pletnev, M. Spaller,
S. Cullati, S. Gerber, P. Boisguerin, D. Casalena, D. Auld, S. Wang, and
D. Madden). 2023 European Cystic Fibrosis Society
Conference. Dubrovnik, Croatia March 29-April 1 2023.
-
Chiral evasion and stereospecific antifolate resistance
in Staphylococcus aureus
(with
S. Wang,
S. Reeve, G. Holt
A. Ojewole,
M. Frenkel,
P. Gainza,
S. Keshpeddy,
V. Fowler, and
D. Wright).
PLoS Computational Biology 2022; 18(2):
e1009855. doi: https://doi.org/10.1371/journal.pcbi.1009855 .
- RESISTOR: An algorithm for predicting resistance mutations using
Pareto optimization over multistate protein design and mutational
signatures (with N. Guerin and T. Kaserer). Proceedings of the
Annual International Conference on Research in Computational
Molecular Biology (RECOMB), San Diego. (May 22-25,
2022). Accepted, In Press.
-
Provable algorithms for
ensemble-based computational protein design and the redesign of
the KRas:RAF-kinase protein:protein interface (with
A. Lowegard, M. Frenkel, J. Jou, A. Ojewole,
and G. Holt).
PLoS Computational Biology 2020;
16(6): e1007447. PMID: 32511232
- Toward Broad Spectrum DHFR inhibitors Targeting Trimethoprim
Resistant Enzymes Identified in Clinical Isolates of
Methicillin-Resistant Staphylococcus aureus. (with
S. Reeve, D. Si, J. Krucinska, Y. Yan, K. Viswanathan, S. Wang,
G. Holt,
M. Frenkel, A. Ojewole, A. Estrada, S. Agabiti, J.
Alverson, N. Gibson, N. Priestly, A. Wiemer, and D. Wright).
ACS
Infectious Diseases
2019; 5(11):1896-1906. .
(doi: 10.1021/acsinfecdis.9b00222)
Preprint on BioRχiv
648808; doi: https://doi.org/10.1101/648808
- Computational Analysis of Energy Landscapes Reveals Dynamic
Features that Contribute to Binding of Inhibitors to CFTR-Associated
Ligand
(with
G. Holt, J. Jou, N. Gill, A. Lowegard,
J. Martin, and D. Madden).
Jour. Physical Chemistry B.
2019; 123(49):10441-10455.
PMID: 31697075
-
T. Kaserer and J. Blagg.
Combining Mutational Signatures, Clonal Fitness, and Drug Affinity to
Define Drug-Specific Resistance Mutations in Cancer.
Cell Chem Biol. 2018; 25(11):1359-1371.e2. doi:
10.1016/j.chembiol.2018.07.013.
- A systematic molecular and pharmacologic evaluation of AKT
inhibitors reveals new insight into their biological activity.
Kostaras E, Kaserer T, Lazaro G, Heuss SF, Hussain A, Casado P, Hayes
A, Yandim C, Palaskas N, Yu Y, Schwartz B, Raynaud F, Chung YL,
Cutillas PR, Vivanco I. Br J Cancer. 2020 May 22. doi:
10.1038/s41416-020-0889-4. Online ahead of print. PMID: 32439931
- Structure-Based Design of a Soluble Prefusion-Closed HIV-1 Env
Trimer with Reduced CD4 Affinity and Improved Immunogenicity. Gwo-Yu
Chuang, Hui Geng, Marie Pancera, Kai Xu, Cheng Cheng, Priyamvada
Acharya, Michael Chambers, Aliaksandr Druz, Yaroslav Tsybovsky,
Timothy G. Wanninger, Yongping Yang, Nicole A. Doria-Rose, Ivelin
S. Georgiev, Jason Gorman, M. Gordon Joyce, Sijy O'Dell, Tongqing
Zhou, Adrian B. McDermott, John R. Mascola, Peter D. Kwong Journal of
Virology Apr 2017, 91 (10) e02268-16; DOI: 10.1128/JVI.02268-16
- S. Reeve, P. Gainza, K. Frey, I. Georgiev, B. R. Donald, and A. Anderson. Protein Design Algorithms
Predict Viable Resistance to an
Experimental Antifolate. Proceedings of the National
Academy of Sciences,
U.S.A. (PNAS). 2015; doi:
10.1073/pnas.1411548112
- R. Rudicell, Y. Kwon, S.Y. Ko,
A. Pegu, M. Louder, I. Georgiev,
X. Wu, J. Zhu, J. Boyington, X. Chen, W. Shi, Z. Yang,
N. Doria-Rose, K. McKee, S. O'Dell, S. Schmidt, G.Y. Chuang, A. Druz,
C. Soto, Y. Yang, B. Zhang, T. Zhou, J.P. Todd, K. Lloyd, J. Eudailey,
K. Roberts,
B. R. Donald, R. Bailer, J. Ledgerwood, NISC
Comparative Sequencing Program, J. Mullikin, L. Shapiro, R. Koup,
B. Graham, M. Nason, M. Connors, B. Haynes, S. Rao, M. Roederer,
P. Kwong, J. Mascola, and G. Nabel.
Enhanced potency of a broadly neutralizing HIV-1 antibody
in vitro improves protection against lentiviral infection
in vivo.
Journal of Virology (2014)
doi: 10.1128/JVI.02213-14
- Ivelin S. Georgiev, Rebecca S. Rudicell, Kevin O. Saunders, Wei
Shi, Tatsiana Kirys, Krisha McKee, Sijy O'Dell, Gwo-Yu Chuang,
Zhi-Yong Yang, Gilad Ofek, Mark Connors, John R. Mascola, Gary
J. Nabel and Peter D. Kwong. Antibodies VRC01 and 10E8 Neutralize
HIV-1 with High Breadth and Potency Even with Ig-Framework Regions
Substantially Reverted to Germline. The Journal of
Immunology (2014). doi:
10.4049/.jimmunol.1302515
- De novo design of a transmembrane Zn2+-transporting four-helix
bundle.
Joh NH, Wang T, Bhate MP, Acharya R, Wu Y, Grabe M, Hong M, Grigoryan
G, DeGrado WF.
Science. 2014 Dec 19;346(6216):1520-4. doi: 10.1126/science.1261172.
PMID: 25525248.
- I. Georgiev, P. Acharya, S. Schmidt, Y. Li, D. Wycuff,
G. Ofek, N. Doria-Rose, T. Luongo, Y, Yang, T. Zhou, B. R. Donald, J.
Mascola, P. Kwong.
Design of Epitope-Specific Probes for Sera Analysis and Antibody
Isolation. Retrovirology 2012;
9(Suppl.2):P50.
- A critical analysis of computational protein design with sparse
residue interaction graphs (with
S. Jain, J. Jou, and I. Georgiev).
PLoS Comput. Biol. 2017 Mar 30;13(3):e1005346. doi:
10.1371/journal.pcbi.1005346.
- Roberts KE, Cushing PR, Boisguerin P, Madden DR, Donald BR. Computational
Design of a PDZ Domain Peptide Inhibitor that Rescues CFTR Activity. PLoS Comput
Biol. 2012 Apr;8(4):e1002477. Epub 2012 Apr 19. PubMed PMID: 22532795; PubMed
Central PMCID: PMC3330111.
- Frey KM, Georgiev I, Donald BR, Anderson AC. Predicting resistance mutations
using protein design algorithms. Proc Natl Acad Sci U S A. 2010 Aug
3;107(31):13707-12. Epub 2010 Jul 19. PubMed PMID: 20643959; PubMed Central
PMCID: PMC2922245.
- Chen CY, Georgiev I, Anderson AC, Donald BR. Computational structure-based
redesign of enzyme activity. Proc Natl Acad Sci U S A. 2009 Mar
10;106(10):3764-9. Epub 2009 Feb 19. PubMed PMID: 19228942; PubMed
Central PMCID: PMC2645347.
- Gorczynski MJ, Grembecka J, Zhou Y, Kong Y, Roudaia L, Douvas MG, Newman M,
Bielnicka I, Baber G, Corpora T, Shi J, Sridharan M, Lilien R, Donald BR, Speck
NA, Brown ML, Bushweller JH. Allosteric inhibition of the protein-protein
interaction between the leukemia-associated proteins Runx1 and CBFbeta. Chem
Biol. 2007 Oct;14(10):1186-97. PubMed PMID: 17961830.
- Stevens BW, Lilien RH, Georgiev I, Donald BR, Anderson AC. Redesigning the
PheA domain of Gramicidin Synthetase leads to a new understanding of the enzyme's
mechanism and selectivity. Biochemistry. 2006 Dec 26;45(51):15495-504. Epub 2006
Dec 19. PubMed PMID: 17176071.
Selected Crystal Stuctures That Confirmed OSPREY Designs:
-
See structures here.
Search
PDB (NCBI) for all our protein structures (NMR, X-ray)
The Book, and Selected Papers on OSPREY Algorithms, Methodology, and Validation:
The textbook describes the algorithms in detail:
Algorithms in Structural Molecular Biology. MIT Press (2011).
Order from Amazon.
- The
most recent algorithms and software papers are here. (MARK*,
CATS, BBK*, EWAK*, FRIES, PPI predictions, etc.)
-
Provable algorithms for
ensemble-based computational protein design and the redesign of
the KRas:RAF-kinase protein:protein interface (with
A. Lowegard, M. Frenkel, J. Jou, A. Ojewole,
and G. Holt).
PLoS Computational Biology 2020;
16(6): e1007447. PMID: 32511232
- M. Hallen, J. Martin, et al.
OSPREY 3.0: Open-Source Protein
Redesign for You, with Powerful New Features.
Journal of Computational Chemistry 2018; 39(30):
2494-2507 Cover article.
Available here:
- M. Hallen, J. Martin, A. Ojewole, J. Jou,
A. Lowegard, M. Frenkel, P. Gainza, H. Nisonoff, A. Mukund, S. Wang,
G. Holt, D. Zhou,
E. Dowd, B. R. Donald*. OSPREY 3.0: Open-Source Protein
Redesign for You, with Powerful New Features. bioRxiv 306324 (Cold
Spring Harbor); doi:
https://doi.org/10.1101/306324. URL:
https://www.biorxiv.org/content/early/2018/04/23/306324.
- Hallen, Mark A. and Bruce R. Donald. "CATS (Coordinates of Atoms by Taylor
Series): Protein design with backbone flexibility in all locally feasible directions."
Bioinformatics 2017;33(14): i5-i12.
- Ojewole, Adegoke A., Jonathan D. Jou, Vance G. Fowler, and Bruce R. Donald. BBK* (Branch and Bound over K*): A Provable and Efficient Ensemble-Based Algorithm to Optimize
Stability and Binding Affinity over Large Sequence Spaces.
Proceedings of the Annual International Conference on Research in Computational Molecular Biology (RECOMB), Hong Kong. (May 3-7,
2017). In: Research in Computational Molecular Biology, Lecture Notes in Computer Science (LNCS), Springer-Verlag (Berlin) vol. 10229, pp. 157-172.
- Hallen, Mark A., Jonathan D. Jou, and Bruce R. Donald.
"LUTE (Local
Unpruned
Tuple Expansion): Accurate continuously flexible protein design with general
energy functions and rigid-rotamer-like efficiency." Research in
Computational Molecular Biology (RECOMB) 2016 proceedings, volume 9649 of Lecture Notes in Computer Science, pp. 122-136. Springer International Publishing, 2016.
- Jou, Jonathan D., Swati Jain, Ivelin S. Georgiev, and Bruce R. Donald. BWM*: A Novel, Provable, Ensemble-based Dynamic Programming Algorithm for Sparse
Approximations of Computational Protein Design.
Proceedings of the Annual International Conference on Research in Computational Molecular Biology (RECOMB), Warsaw, April 12-15, 2015. In Research in
Computational Molecular Biology Lecture Notes in Computer Science, Springer-Verlag (Berlin), Volume 9029, 2015, pp 154-166
- Hallen, Mark A., Pablo Gainza, and Bruce R. Donald.
"Compact
representation of continuous energy surfaces for more efficient protein
design." Journal of Chemical Theory and Computation 2015;11(5):2292-2306.
- Hallen, Mark A. and Bruce R. Donald.
"COMETS (Constrained Optimization of
Multistate Energies by Tree Search): A provable and efficient algorithm to
optimize binding affinity and specificity with respect to
sequence."
Research in Computational Molecular Biology (RECOMB) 2015 proceedings,
volume 9029 of Lecture Notes in Computer Science, pp. 122-135. Springer
International Publishing, 2015.
-
P. Gainza, K. Roberts, I. Georgiev, R. Lilien, D. Keedy, C.-Y. Chen, F. Reza,
A Anderson, D. Richardson, J. Richardson, and B. R. Donald.
OSPREY: Protein design with ensembles, flexibility, and provable algorithms.
Methods in Enzymology, Vol. 523, Methods in Protein Design, pp87-107. (2013).
ISBN: 9780123942920.
http://store.elsevier.com/Methods-in-Protein-Design/isbn-9780123942920/
- Structure-guided deimmunization of therapeutic proteins.
Parker AS, Choi Y, Griswold KE, Bailey-Kellogg C.
J Comput Biol. 2013 Feb;20(2):152-65. doi: 10.1089/cmb.2012.0251.
- Hallen MA, Keedy DA, Donald BR. Dead-End Elimination with Perturbations
(DEEPer): A Provable Protein Design Algorithm with Continuous Sidechain and
Backbone Flexibility. Proteins. 2012, in press. Epub 2012 Jul 21. PubMed PMID:
22821798.
- Y. Zhou, W. Xu, B. R. Donald,
and J. (Michael)
Zeng. An efficient parallel algorithm for accelerating
computational protein design.
Bioinformatics. 2014 Jun 15;30(12):i255-i263. Proceedings
of ISMB, Boston, MA. doi: 10.1093/bioinformatics/btu264.
- Roberts KE, Cushing PR, Boisguerin P, Madden DR, Donald BR. Computational
Design of a PDZ Domain Peptide Inhibitor that Rescues CFTR Activity. PLoS Comput
Biol. 2012 Apr;8(4):e1002477. Epub 2012 Apr 19. PubMed PMID: 22532795; PubMed
Central PMCID: PMC3330111.
- Gainza P, Roberts KE, Donald BR. Protein design using continuous rotamers.
PLoS Comput Biol. 2012 Jan;8(1):e1002335. Epub 2012 Jan 12. PubMed PMID:
22279426; PubMed Central PMCID: PMC3257257.
- Frey KM, Georgiev I, Donald BR, Anderson AC. Predicting resistance mutations
using protein design algorithms. Proc Natl Acad Sci U S A. 2010 Aug
3;107(31):13707-12. Epub 2010 Jul 19. PubMed PMID: 20643959; PubMed Central
PMCID: PMC2922245.
- Chen CY, Georgiev I, Anderson AC, Donald BR. Computational structure-based
redesign of enzyme activity. Proc Natl Acad Sci U S A. 2009 Mar
10;106(10):3764-9. Epub 2009 Feb 19. PubMed PMID: 19228942; PubMed Central PMCID: PMC2645347.
- Georgiev I, Keedy D, Richardson JS, Richardson DC, Donald BR. Algorithm for
backrub motions in protein design. Bioinformatics. 2008 Jul 1;24(13):i196-204.
PubMed PMID: 18586714; PubMed Central PMCID: PMC2718647.
- Georgiev I, Donald BR. Dead-end elimination with backbone flexibility.
Bioinformatics. 2007 Jul 1;23(13):i185-94. PubMed PMID: 17646295.
- Georgiev I, Lilien RH, Donald BR. The minimized dead-end elimination criterion
and its application to protein redesign in a hybrid scoring and search algorithm
for computing partition functions over molecular ensembles. J Comput Chem. 2008
Jul 30;29(10):1527-42. PubMed PMID: 18293294; PubMed Central PMCID: PMC3263346.
- Lilien RH, Stevens BW, Anderson AC, Donald BR. A novel ensemble-based scoring
and search algorithm for protein redesign and its application to modify the
substrate specificity of the Gramicidin Synthetase A phenylalanine adenylation
enzyme. J Comput Biol. 2005 Jul-Aug;12(6):740-61. PubMed PMID: 16108714.
- Georgiev I, Lilien RH, Donald BR. Improved Pruning algorithms and
Divide-and-Conquer strategies for Dead-End Elimination, with application to
protein design. Bioinformatics. 2006 Jul 15;22(14):e174-83. PubMed PMID:
16873469.